E. Kostenis: search on Z-Library

The world's largest scientific articles store. 70,000,000+ articles for free.

Don't use scam websites

1

Author Correction: Chemokine receptor trafficking coordinates neutrophil clustering and dispersal at wounds in zebrafish

Coombs, Caroline, Georgantzoglou, Antonios, Walker, Hazel A., Patt, Julian, Merten, Nicole, Poplimont, Hugo, Busch-Nentwich, Elisabeth M., Williams, Sarah, Kotsi, Christina, Kostenis, Evi, Sarris, Mil

Journal:

Nature Communications

Year:

2020

Language:

english

File:

PDF, 408 KB

english, 2020

2

G q/11 -dependent regulation of endosomal cAMP generation by parathyroid hormone class B GPCR

White, Alex D., Jean-Alphonse, Frederic G., Fang, Fei, PeÃ±a, Karina A., Liu, Shi, KÃ¶nig, Gabriele M., Inoue, Asuka, Aslanoglou, Despoina, Gellman, Samuel H., Kostenis, Evi, Xiao, Kunhong, Vilardaga,

Journal:

Proceedings of the National Academy of Sciences

Year:

2020

Language:

english

File:

PDF, 1.46 MB

english, 2020

3

Functional selectivity and dualsteric/bitopic GPCR targeting

Schrage, Ramona, Kostenis, Evi

Journal:

Current Opinion in Pharmacology

Year:

2017

Language:

english

File:

PDF, 377 KB

english, 2017

4

Veranstaltungen 2014

Teutsch, Charlott-Amelie, Panse, Madhura, Grundmann, Manuel, Kaiser, Gabriele, Kostenis, Evi, Häring, Hans-Ulrich, Ullrich, Susanne

Journal:

Zeitschrift für Energiewirtschaft

Year:

2014

File:

PDF, 59 KB

2014

5

Novel selective thiazoleacetic acids as CRTH2 antagonists developed from in silico derived hits. Part 1

Øystein Rist, Marie Grimstrup, Jean-Marie Receveur, Thomas M. Frimurer, Trond Ulven, Evi Kostenis, Thomas Högberg

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2010

Language:

english

File:

PDF, 420 KB

english, 2010

6

Rational design of dualsteric GPCR ligands: quests and promise

Klaus Mohr, Christian Tränkle, Evi Kostenis, Elisabetta Barocelli, Marco De Amici, Ulrike Holzgrabe

Journal:

British Journal of Pharmacology

Year:

2010

Language:

english

File:

PDF, 519 KB

english, 2010

7

β-Arrestin 2 Inhibits Proinflammatory Chemokine Production and Attenuates Contact Allergic Inflammation in the Skin

Gaffal, Evelyn, Jakobs, Mira, Glodde, Nicole, Schröder, Ralf, Kostenis, Evi, Tüting, Thomas

Journal:

The Journal of Investigative Dermatology

Year:

2014

Language:

english

File:

PDF, 6.08 MB

english, 2014

8

Reactivation of Gαi-coupled formyl peptide receptors is inhibited by Gαq-selective inhibitors when induced by signals generated by the platelet-activating factor receptor

Holdfeldt, André, Dahlstrand Rudin, Agnes, Gabl, Michael, Rajabkhani, Zahra, König, Gabriele M., Kostenis, Evi, Dahlgren, Claes, Forsman, Huamei

Journal:

Journal of Leukocyte Biology

Year:

2017

Language:

english

File:

PDF, 1.32 MB

english, 2017

9

Pronounced pharmacologic deficits in M2 muscarinic acetylcholine receptor knockout mice

Gomeza, J., Shannon, H., Kostenis, E., Felder, C., Zhang, L., Brodkin, J., Grinberg, A., Sheng, H., Wess, J.

Journal:

Proceedings of the National Academy of Sciences

Year:

1999

Language:

english

File:

PDF, 199 KB

english, 1999

10

Extracellular Loop 2 of the Free Fatty Acid Receptor 2 Mediates Allosterism of a Phenylacetamide Ago-Allosteric Modulator

Smith, N. J., Ward, R. J., Stoddart, L. A., Hudson, B. D., Kostenis, E., Ulven, T., Morris, J. C., Trankle, C., Tikhonova, I. G., Adams, D. R., Milligan, G.

Journal:

Molecular Pharmacology

Year:

2011

Language:

english

File:

PDF, 2.33 MB

english, 2011

11

Functional Human 5-HT6 Receptor Assay for High Throughput Screening of Chemical Ligands and Binding Proteins

Kim, Hyun-Ji, Yun, Hyung-Mun, Kim, Taehyun, Nam, Ghilsoo, Roh, Eun, Kostenis, Evi, Choo, Hea-Young, Pae, Ae, Rhim, Hyewhon

Journal:

Combinatorial Chemistry & High Throughput Screening

Year:

2008

Language:

english

File:

PDF, 446 KB

english, 2008

12

Temporal Bias: Time-Encoded Dynamic GPCR Signaling

Grundmann, Manuel, Kostenis, Evi

Journal:

Trends in Pharmacological Sciences

Year:

2017

Language:

english

File:

PDF, 2.86 MB

english, 2017

13

Novel selective thiazoleacetic acids as CRTH2 antagonists developed from in silico derived hits. Part 2

Marie Grimstrup, Øystein Rist, Jean-Marie Receveur, Thomas M. Frimurer, Trond Ulven, Jesper M. Mathiesen, Evi Kostenis, Thomas Högberg

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2010

Language:

english

File:

PDF, 1.52 MB

english, 2010

14

The D-type prostanoid (DP) receptor enhances the signaling of chemoattractant receptor-homologous molecule expressed on Th2 cells (CRTH2)

Miriam Sedej, Ralf Schröder, Kathrin Bell, Wolfgang Platzer, Evi Kostenis, Ákos Heinemann, Maria Waldhoer

Journal:

BMC Pharmacology

Year:

2011

Language:

english

File:

PDF, 64 KB

english, 2011

15

Enhancement of D1 dopamine receptor-mediated locomotor stimulation in M4 muscarinic acetylcholine receptor knockout mice

Gomeza, J., Zhang, L., Kostenis, E., Felder, C., Bymaster, F., Brodkin, J., Shannon, H., Xia, B., Deng, C.-x., Wess, J.

Journal:

Proceedings of the National Academy of Sciences

Year:

1999

Language:

english

File:

PDF, 166 KB

english, 1999

16

Heterotrimeric Gq proteins as therapeutic targets?

Kostenis, Evi, Pfeil, Eva Marie, Annala, Suvi

Journal:

Journal of Biological Chemistry

Year:

2020

File:

PDF, 1.01 MB

2020

17

FFA2-, but not FFA3-agonists inhibit GSIS of human pseudoislets: a comparative study with mouse islets and rat INS-1E cells

Lorza-Gil, Estela, Kaiser, Gabriele, Rexen Ulven, Elisabeth, KÃ¶nig, Gabriele M., Gerst, Felicia, Oquendo, Morgana Barroso, Birkenfeld, Andreas L., HÃ¤ring, Hans-Ulrich, Kostenis, Evi, Ulven, Trond, U

Journal:

Scientific Reports

Year:

2020

File:

PDF, 1.59 MB

2020

18

Functional expression of M1, M3 and M5 muscarinic acetylcholine receptors in yeast

Isolde Erlenbach, Evi Kostenis, Clarice Schmidt, Fadi F. Hamdan, Mark H. Pausch, Jürgen Wess

Journal:

Journal of Neurochemistry

Year:

2001

Language:

english

File:

PDF, 773 KB

english, 2001

19

The β2-subtype of adrenoceptors mediates inhibition of pro-fibrotic events in human lung fibroblasts

F. Lamyel, M. Warnken-Uhlich, W. K. Seemann, K. Mohr, E. Kostenis, A. S. Ahmedat, M. Smit, R. Gosens, H. Meurs, A. Miller-Larsson, Kurt Racké

Journal:

Naunyn-Schmiedeberg's Archives of Pharmacology

Year:

2011

Language:

english

File:

PDF, 534 KB

english, 2011

20

Structure-function analysis of muscarinic receptors and their associated G proteins

Evi Kostenis, Fu-Yue Zeng, Jürgen Wess

Journal:

Year:

1999

Language:

english

File:

PDF, 733 KB

english, 1999

21

Identification of a Potent and Selective Free Fatty Acid Receptor 1 (FFA1/GPR40) Agonist with Favorable Physicochemical and in Vitro ADME Properties

Christiansen, Elisabeth, Urban, Christian, Grundmann, Manuel, Due-Hansen, Maria E., Hagesaether, Ellen, Schmidt, Johannes, Pardo, Leonardo, Ullrich, Susanne, Kostenis, Evi, Kassack, Matthias, Ulven, T

Journal:

Journal of Medicinal Chemistry

Year:

2011

Language:

english

File:

PDF, 3.65 MB

english, 2011

22

Molecular Basis of Receptor/G Protein Coupling Selectivity Studied by Coexpression of Wild Type and Mutant m2 Muscarinic Receptors with Mutant Gα q Subunits †

Kostenis, Evi, Conklin, Bruce R., Wess, Jürgen

Journal:

Year:

1997

Language:

english

File:

PDF, 194 KB

english, 1997

23

G Proteins in Drug Screening: From Analysis of Receptor-G Protein Specificity to Manipulation of GPCR-Mediated Signalling Pathways

Journal:

Current Pharmaceutical Design

Year:

2006

Language:

english

File:

PDF, 249 KB

english, 2006

24

Gβγ signaling to the chemotactic effector P-REX1 and mammalian cell migration is directly regulated by Gαq and Gα13 proteins

Cervantes-Villagrana, Rodolfo Daniel, Adame-García, Sendi Rafael, García-Jimenez, Irving, Color-Aparicio, Víctor Manuel, Beltran-Navarro, Yarely Mabell, König, Gabriele M., Kostenis, Evi, Reyes-Cruz,

Journal:

Journal of Biological Chemistry

Year:

2018

Language:

english

File:

PDF, 2.34 MB

english, 2018

25

Probing Allosteric Binding Site Mapping in the Free Fatty Acid 2 receptor

Tikhonova, Irina G., Smith, Nicola J., Ward, Richard J., Stoddart, Leigh A., Hudson, Brian D., Kostenis, Evi, Ulven, Trond, Morris, Joanne C., Adams, David R., Milligan, Graeme

Journal:

Biophysical Journal

Year:

2011

Language:

english

File:

PDF, 35 KB

english, 2011

26

D-type prostanoid receptor enhances the signaling of chemoattractant receptor–homologous molecule expressed on TH2 cells

Sedej, Miriam, Schröder, Ralf, Bell, Kathrin, Platzer, Wolfgang, Vukoja, Anela, Kostenis, Evi, Heinemann, Akos, Waldhoer, Maria

Journal:

Journal of Allergy and Clinical Immunology

Year:

2012

Language:

english

File:

PDF, 1.85 MB

english, 2012

27

POTENTIATION OF GPCR-SIGNALING VIA MEMBRANE TARGETING OF G PROTEIN α SUBUNITS

Journal:

Journal of Receptor and Signal Transduction Research

Year:

2002

Language:

english

File:

PDF, 395 KB

english, 2002

28

A Molecular Mechanism for Sequential Activation of a G Protein-Coupled Receptor

Grundmann, Manuel, Tikhonova, Irina G., Hudson, Brian D., Smith, Nicola J., Mohr, Klaus, Ulven, Trond, Milligan, Graeme, Kenakin, Terry, Kostenis, Evi

Journal:

Cell Chemical Biology

Year:

2016

Language:

english

File:

PDF, 3.28 MB

english, 2016

29

cNMP-AMs mimic and dissect bacterial nucleotidyl cyclase toxin effects

Beckert, Ulrike, Grundmann, Manuel, Wolter, Sabine, Schwede, Frank, Rehmann, Holger, Kaever, Volkhard, Kostenis, Evi, Seifert, Roland

Journal:

Biochemical and Biophysical Research Communications

Year:

2014

Language:

english

File:

PDF, 1.01 MB

english, 2014

30

The molecular mechanism by which saturated lysophosphatidylcholine attenuates the metastatic capacity of melanoma cells

Ross, Thomas, Jakubzig, Bastian, Grundmann, Manuel, Massing, Ulrich, Kostenis, Evi, Schlesinger, Martin, Bendas, Gerd

Journal:

Year:

2016

Language:

english

File:

PDF, 1.19 MB

english, 2016

31

Bruton's Tyrosine Kinase and RAC1 promote cell survival in MLL-rearranged acute myeloid leukemia

Nimmagadda, S C, Frey, S, Edelmann, B, Hellmich, C, Zaitseva, L, König, G M, Kostenis, E, Bowles, K M, Fischer, T

Journal:

Year:

2017

Language:

english

File:

PDF, 1.72 MB

english, 2017

32

Applying Molecular Networking for the Detection of Natural Sources and Analogues of the Selective Gq Protein Inhibitor FR900359

Reher, Raphael, Kuschak, Markus, Heycke, Nina, Annala, Suvi, Kehraus, Stefan, Dai, Hao-Fu, Müller, Christa E., Kostenis, Evi, König, Gabriele M., Crüsemann, Max

Journal:

Journal of Natural Products

Year:

2018

Language:

english

File:

PDF, 1.91 MB

english, 2018

33

Biased signaling of Ca2+-sensing receptors in cardiac myocytes regulates GIRK channel activity

Kienitz, Marie-Cecile, Niemeyer, Anne, König, Gabriele M., Kostenis, Evi, Pott, Lutz, Rinne, Andreas

Journal:

Journal of Molecular and Cellular Cardiology

Year:

2019

Language:

english

File:

PDF, 2.15 MB

english, 2019

34

Exploring Biased Agonism at FPR1 as a Means to Encode Danger Sensing

GrÃ¶per, Jieny, KÃ¶nig, Gabriele M., Kostenis, Evi, Gerke, Volker, Raabe, Carsten A., Rescher, Ursula

Journal:

Year:

2020

File:

PDF, 4.26 MB

2020

35

Tetrahydroimidazo[1,2âa]pyrazine Derivatives: Synthesis and Evaluation As GÎ±qâProtein Ligands

GÃ¼tschow, Michael, KÃ¼ppers, Jim, Benkel, Tobias, Annala, Suvi, Kimura, Kenichi, Reinelt, Lisa, Fleischmann, Bernd K., Kostenis, Evi

Journal:

Chemistry (Weinheim an der Bergstrasse, Germany)

Year:

2020

File:

PDF, 1.14 MB

2020

36

Kostenis and Mohr reply: Composite action of allosteric modulators on ligand binding

Evi Kostenis, Klaus Mohr

Journal:

Trends in Pharmacological Sciences

Year:

1996

Language:

english

File:

PDF, 259 KB

english, 1996

37

Pro-fibrotic processes in human lung fibroblasts are driven by an autocrine/paracrine endothelinergic system

Ahmedat, AS, Warnken, M, Seemann, WK, Mohr, K, Kostenis, E, Juergens, UR, Racké, K

Journal:

British Journal of Pharmacology

Year:

2013

Language:

english

File:

PDF, 3.47 MB

english, 2013

38

A Biased Non-G i OXE-R Antagonist Demonstrates That G i Protein Subunit Is Not Directly Involved in Neutrophil, Eosinophil, and Monocyte Activation by 5-Oxo-ETE

Konya, V., Blattermann, S., Jandl, K., Platzer, W., Ottersbach, P. A., Marsche, G., Gutschow, M., Kostenis, E., Heinemann, A.

Journal:

The Journal of Immunology

Year:

2014

Language:

english

File:

PDF, 1.73 MB

english, 2014

39

Heterotrimeric G-proteins: a short history

Graeme Milligan, Evi Kostenis

Journal:

British Journal of Pharmacology

Year:

2006

Language:

english

File:

PDF, 269 KB

english, 2006

40

Novel Insights Into Appropriate Encapsulation Methods for Bioactive Compounds Into Polymers: A Study With Peptides and HDAC Inhibitors

Hennig, Dorle, Schubert, Stephanie, Dargatz, Harald, Kostenis, Evi, Fahr, Alfred, Schubert, Ulrich S., Heinzel, Thorsten, Imhof, Diana

Journal:

Macromolecular Bioscience

Year:

2014

Language:

english

File:

PDF, 573 KB

english, 2014

41

P78 potentiation by alcuronium of the antimuscarinic effect on N-methyl-scoplamine in guinea pig left atrium

Maaβ, A., Kostenis, E., Tränkle, C., Mohr, K.

Journal:

European Journal of Pharmaceutical Sciences

Year:

1994

Language:

english

File:

PDF, 122 KB

english, 1994

42

GPR55: signaling pathways and functions

Nariman Balenga, Ralf Schröder, Julia Kargl, Wolfgang Platzer, Stefanie Blättermann, Ákos Heinemann, Evi Kostenis, Maria Waldhoer

Journal:

BMC Pharmacology

Year:

2009

Language:

english

File:

PDF, 72 KB

english, 2009

43

A glance at G-protein-coupled receptors for lipid mediators: a growing receptor family with remarkably diverse ligands

Journal:

Pharmacology & Therapeutics

Year:

2004

Language:

english

File:

PDF, 355 KB

english, 2004

44

Potentiation by alcuronium of the antimuscarinic effect of N-methylscopolamine in guinea pig left atria

Andrea Maaß, Evi Kostenis, Klaus Mohr

Journal:

European Journal of Pharmacology

Year:

1995

Language:

english

File:

PDF, 506 KB

english, 1995

45

Synthesis and in vitro evaluation of a selective antagonist and the corresponding radioligand for the prostaglandin D2 receptor CRTH2

Trond Ulven, Michael J. Gallen, Mads C. Nielsen, Nicole Merten, Carola Schmidt, Klaus Mohr, Christian Tränkle, Evi Kostenis

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2007

Language:

english

File:

PDF, 177 KB

english, 2007

46

Signalling and function of the human G protein-coupled receptor 55

Nariman Balenga, Julia Kargl, Ralf Schröder, Ákos Heinemann, Evi Kostenis, Maria Waldhoer

Journal:

BMC Pharmacology

Year:

2010

Language:

english

File:

PDF, 132 KB

english, 2010

47

Chemically engineering ligand selectivity at the free fatty acid receptor 2 based on pharmacological variation between species orthologs

Hudson, B. D., Christiansen, E., Tikhonova, I. G., Grundmann, M., Kostenis, E., Adams, D. R., Ulven, T., Milligan, G.

Journal:

The FASEB Journal

Year:

2012

Language:

english

File:

PDF, 1.02 MB

english, 2012

48

Enhancement of D1 Dopamine Receptor-Mediated Locomotor Stimulation in M4Muscarinic Acetylcholine Receptor Knockout Mice

Jesus Gomeza, Lu Zhang, Evi Kostenis, Christian Felder, Frank Bymaster, Jesse Brodkin, Harlan Shannon, Bing Xia, Chu-xia Deng and Jurgen Wess

Journal:

Proceedings of the National Academy of Sciences

Year:

1999

Language:

english

File:

PDF, 1.60 MB

english, 1999

49

Identification of Nonpeptidic Urotensin II Receptor Antagonists by Virtual Screening Based on a Pharmacophore Model Derived from Structure−Activity Relationships and Nuclear Magnetic Resonance Studies on Urotensin II

Flohr, Stefanie, Kurz, Michael, Kostenis, Evi, Brkovich, Alexandre, Fournier, Alain, Klabunde, Thomas

Journal:

Journal of Medicinal Chemistry

Year:

2002

Language:

english

File:

PDF, 355 KB

english, 2002

50

Dualsteric GPCR targeting: a novel route to binding and signaling pathway selectivity

Antony, J., Kellershohn, K., Mohr-Andra, M., Kebig, A., Prilla, S., Muth, M., Heller, E., Disingrini, T., Dallanoce, C., Bertoni, S., Schrobang, J., Trankle, C., Kostenis, E., Christopoulos, A., Holtj

Journal:

The FASEB Journal

Year:

2008

Language:

english

File:

PDF, 357 KB

english, 2008

To build up a library is to create a life. It’s never just a random collection of books.

— Carlos María Domínguez

Official channel

Z-Library Desktop Launcher

Z-Library Since 2009 support@1delivery.pm

EnglishРусскийEspañolItalianoελληνικάاللغة العربيةBahasa IndonesiaBahasa Malaysiaहिन्दीDeutschFrançaisPortuguêsУкраїнськаPolski中文繁體中文日本語Tiếng ViệtAzərbaycan DiliՀայոց լեզուภาษาไทยTürk Diliქართველიবাংলাپښتوతెలుగుاردو한국어SrpskiБългарски